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发表论文Publications

Mesoporous carbon hemispheres integrated with Fe–Gd nanoparticles for potential MR/PA imaging-guided photothermal therapy Mengmeng Zhang, Tianze Wu, Hui Zhang, Zhenxia Chen,  Yannan Yang, Yun Ling * and Yaming Zhou,*  Journal of Materials Chemistry B2024, 12, 658-666 >> Fulltext link

Systematical Evaluation of the Structure-Cardiotoxicity Relationship of 7-Azaindazole-based PI3K Inhibitors Designed by Bioisosteric Approach Tianze Wu, Yi Chen, Chengbin Yang, Mingzhu Lu, Fang Geng, Jianhua Guo, Yan Pi, Yun Ling, Jun Xu, Tong Cai, Lei Lu & Yaming Zhou,*  Cardiovascular Toxicology2023, 23, 364-376 >> Fulltext link

Discovery and identification of a novel PI3K inhibitor with enhanced CDK2 inhibition for the treatment of triple negative breast cancer Chengbin Yang, Menghui Wang, Yimin Gong, Mingli Deng, Yun Ling, Qingquan Li, Jianxin Wang*, Yaming Zhou,*  Bioorganic Chemistry2023, 140, 106779 >> Fulltext link

Discovery of a photosensitizing PI3K inhibitor for tumor therapy: Design, synthesis and in vitro biological evaluation Chengbin Yang, Yimin Gong, Mingli Deng, Yun Ling, Jianxin Wang*, Yaming Zhou,*  Bioorganic & Medicinal Chemistry Letters2023,94, 129459 >> Fulltext link


Reticular chemistry of the fcu-type Gd(III)-doped metal-organic framework for T1-weighted magnetic resonance imaging,Tianze Qiu; Tianze Wu; Mingzhu Lu; Yuxi Xie; Mengmeng Zhang; Dan Luo; Zhenxia Chen; Bo Yin; Yaming Zhou; Yun Ling,*  Small2023, 2303063 >> Fulltext link

Discovery of N-(2-chloro-5-(3-(pyridin-4-yl)-1H-pyrazolo[3,4-b]pyridin-5-yl)pyridin-3-yl)-4-fluorobenzenesulfonamide (FD274) as a highly potent PI3K/mTOR dual inhibitor for the treatment of acute myeloid leukemia Chengbin Yang, Yi Chen, Tianze Wu, Yunjian Gao, Xiaofeng Liu, Yongtai Yang, Yun Ling, Yu Jia, Mingli Deng*, Jianxin Wang, Yaming Zhou,*  European Journal of Medicinal Chemistry2023, 258, 115543 >> Fulltext link

Nanosheets of two-dimensional photoluminescent Lanthanide phosphonocarboxylate frameworks decorated with free carboxylic groups for latent fingerprint imaging Dan Luo,   Hongjie He,   Huiru Jing,   Yun Ling,   Yu Jia,   Yongtai Yang,   Xiaofeng Liu,   Zhenxia Chen*  and  Mingli Deng*   Dalton Transcations2023, 52, 9208-9214;>> Fulltext link

Gelothermal Synthesis of Monodisperse MIL-88A Nanoparticles with Tunable Sizes and Metal Centers for Potential Bioapplications Mengmeng Zhang, Mingzhu Lu, Tianze Qiu, Qiao Wang, Zhenxia Chen, Mingli Deng, Yongtai Yang, Yannan Yang, Wei Li, Yun Ling,* and Yaming Zhou  Small2023, 19(34), 2301894 >> Fulltext link

Discovery of a high potent PIM kinase inhibitor for acute myeloid leukemia based on N-pyridinyl amide scaffold by optimizing the fragments toward to Lys67 and Asp128/Glu171 Ruiqing Xiang, Mingzhu Lu, Tianze Wu, Chengbin Yang, Yu Jia,  Xiaofeng Liu, Mingli Deng,**, Yu Ge, Jun Xu, Tong Cai, Yun Ling, Yaming Zhou,*  European Journal of Medicinal Chemistry2023, 223, 257, 115514 >> Fulltext link

Design, synthesis and in vitro biological evaluation of 2-aminopyridine derivatives as novel PI3Kδ inhibitors for hematological cancerChengbin Yang, Yimin Gong, Yunjian Gao, Mingli Deng,  Xiaofeng Liu, Yongtai Yang, Yun Ling, Yu Jia*, Yaming Zhou*; Bioorg. Med. Chem. Lett.2023, 82, 129152>> Fulltext link


Gadolinium-based contrast agents built of DO3A-pyridine scaffold: Precisely tuning carboxylate group for enhanced magnetic resonance imagingYongyin Geng, TianzeWu, Qiuyue Han, Yongtai Yang, Zhenxia Chen, Xuanxuan Li, Bo Yin, Yaming Zhou, Yun Ling*; Chinese Chemical Letters2023, 34, 107685>> Fulltext link


A Pyridinesulfonamide Derivative FD268 Suppresses Cell Proliferation and Induces Apoptosis via Inhibiting PI3K Pathway in Acute Myeloid LeukemiaYi Chen,  Tianze Wu, Chengbin Yang, Mingzhu Lu, Zhenxia Chen, Mingli Deng, Yu Jia, Yongtai Yang, Xiaofeng Liu,  Hongyan Wang, Yun Ling,, Lei Lu,* Yaming Zhou*; PLoS ONE2022, 17(11):e0277893>> Fulltext link

Hybrid Nanomaterials for Cancer ImmunotherapyJianing Li, Wanyue Lu, Yannan Yang*, Ruiqing Xiang, Yun Ling, Chengzhong Yu*, Yaming Zhou*; Advanced Science2022, 2204932>> Fulltext link

Physical and Chemical Cues at the Nano–Bio Interface for ImmunomodulationFeng-Yuan Wang, Tianze Qiu, Yun Ling, Yannan Yang,* and Yaming Zhou*; Angew. Chem. Int. Ed. 2022, 61, e202209499>> Fulltext link


Unprecedented Ferromagnetic Exchange Coupling of a Square-Planar Cu4O unit in a scu-Type Porous Metal–Organic Framework and Its Reticular ChemistryTianze Qiu, Yongchen Wang, Yihan Li, Lin Zhu*, Zhenxia Chen, Yu Jia, Pu Zhao, Wei Shi, Yaming Zhou, and Yun Ling*; Cryst. Growth Des.2022, 22, 7, 4005–4011>> Fulltext link

Hollow carbon nanospheres embedded with stoichiometric γ-Fe2O3 and GdPO4: tuning the nanospheres for in vitro and in vivo size effect evaluation, Hui Zhang,   Jianping Zhang,   Yi Chen,   Tianze Wu,   Mingzhu Lu,   Zhenxia Chen, Yu Jia,   Yongtai Yang,  Yun Ling*  and  Yaming Zhou*; Nanoscale Advances2022, 4, 1414 >> Fulltext link

Development of Anti-Breast Cancer PI3K Inhibitors Based on 7-Azaindole Derivatives through Scaffold Hopping: Design, Synthesis and in Vitro Biological Evaluation, Chengbin Yang, Mingzhu Lu, Yi Chen, Ruiqing Xiang, Tianze Qiu, Yu Jia, Yongtai Yang, Xiaofeng Liu, Mingli Deng, Yun Ling, Yaming Zhou*; Bioorganic Chemistry2021, 117, 105405 >> Fulltext link

Ultrafine Fe-modulated Ni nanoparticles embedded within nitrogen-doped carbon from Zr-MOFs-confined conversion for efficient oxygen evolution reaction, Lingtao Kong, Zhouxun Li, Hui Zhang, Mengmeng Zhang, Jiaxing Zhu, Mingli Deng*, Zhenxia Chen, Yun Ling & Yaming Zhou, Frontiers of Chemical Science and Engineering2022, 16, 1114–1124  >> Fulltext link

Effect of Fluorination on the Crystal Structure, Stability and Gas Adsorption Property in Zinc(II) Metal-organic Frameworks, Xin Zhang, Zhenxia Chen, Yongtai Yang, Mingli Deng*, Linhong Weng; Chinese Journal of Structrual Chemistry2022, 41(2), 49-56 >> Fulltext link

Post-synthetic anchoring Fe(III) into a fcu-type Zr-MOF for the catalyzed hydrolysis of 5-hydroxylmethoxyfurfural, Mengmeng Zhang, Jiaying Lou, Rui Xu, Peng Li, Yunfei Sha, Hui Zhang, Yu Jia, Zhenxia Chen, Da Wu*, Yun Ling*, YamingZhou; Microporous Mesoporous Materials2021, 328, 111449 >> Fulltext link



Reticular Chemistry Approach to Explore the Catalytic CO2-epoxide Cycloaddition Reaction over Tetrahedral Coordination Lewis Acidic Sites in a Rutile-type Zinc-phosphonocarboxylate FrameworkLingtao Kong, Zhouxun Li, Han Hu, Jiaxing Zhu, Zhenxia Chen*, Mingli Deng*, Yun Ling, Peng Li, Yu Jia, Yaming Zhou;  Chemical Engineering Journal2022, 427,131759 >> Fulltext link 


Discovery of cinnoline derivatives as potent PI3K inhibitors with antiproliferative activityChengze Tian, Chengbin Yang, Tianze Wu, Mingzhu Lu, Yi Chen, Yongtai Yang, Xiaofeng Liu, Yun Ling, Mingli Deng, Yu Jia*, Yaming Zhou*  Bioorganic & Medicinal Chemistry Letters2021, 48, 128271 >> Fulltext link


Bioisosteric replacements of the indole moiety for the development of a potent and selective PI3Kδ inhibitor: Design, synthesis and biological evaluationChengbin Yang, Chenyue Xu, Zhipeng Li, Yi Chen, Tianze Wu, Hui Hong, Mingzhu Lu, Yu Jia, Yongtai Yang, Xiaofeng Liu, Mingli Deng, Zhenxia Chen, Qingquan Li*, Yun Ling*, Yaming Zhou*  European Journal of Medicinal Chemistry2021, 223, 1136613 >> Fulltext link


Hollow carbon nanospheres dotted with Gd–Fe nanoparticles for magnetic resonance and photoacoustic imagingHui Zhang,  Tianze Wu, Yi Chen, Qianqian Zhang, Zhenxia Chen,  Yun Ling,* Yu Jia,   Yongtai Yang,   Xiaofeng Liu  and Yaming Zhou*  Nanaoscale2021, 13, 10943-10952 >> Fulltext link


Multimetal lanthanide phosphonocarboxylate frameworks: structure, colour tuning and near-infrared emissionHuiru Jing,   Wenyan Dan,   Jiaxing Zhu,   Yun Ling,   Yu Jia,   Yongtai Yang,   Xiaofeng Liu,   Zhenxia Chen*  and  Yaming Zhou*  Dalton Transcations2021, 50, 7380 - 7387 >> Fulltext link


TEA-assistant synthesis of MOF-74 nanorods for drug delivery and in-vitro magnetic resonance imagingJiaqi Hu, Yi Chen, Hui Zhang, Zhenxia Chen*, Yun Ling, Yongtai Yang, Xiaofeng Liu, Yu Jia, Yaming ZhouMicroporous Mesoporous Materials2021, 315, 110900 >> Fulltext link

  

 

Controlled syntheses of Mg-MOF-74 nanorods for Drug DeliveryJiaqi Hu; Yi Chen; Hui Zhang; Zhenxia Chen*, Journal of Solid State Chemistry2021, 294, 121853 >> Fulltext link


Precise regulating synergistic effect in metal–organic framework for stepwise-controlled adsorptionJiaxing Zhu, Yi Yu, Hongchuan Fan, Huaqiang Cai,*  Zhenxia Chen,  Linhong Weng,  Yun Ling*  and  Yaming ZhouInorganic Chemistry Frontier2021, 8, 1666-1674 >> Fulltext link

In situ embedding dual-Fe nanoparticles in synchronously generated carbon for the synergistic integration of magnetic resonance imaging and drug deliveryHui Zhang; Jianping Zhang; Qianqian Zhang; Xiaofeng Liu; Yongtai Yang; Yun Ling; Yaming Zhou*Nanoscale Advances2020,2, 5296-5304 >> Fulltext link

Coordination and space confined preparation of nickel sub-nanoparticles within a metal-organic framework for catalytic degradation of methyl orangeZhouxun Li, Hui Zhang, Lingtao Kong, Zhenxia Chen*, Yongtai Yang, Xiaofeng Liu, Mingli Deng*, Yaming Zhou, Journal of Environmental Chemical Engineering2020,8(5),104363 >> Fulltext link


Cobalt substitution in a flexible metal-organic framework: modulating a soft paddle-wheel unit for tunable gate-opening adsorptionJiaxing Zhu; Junye Chen; Tianze Qiu; Mingli Deng*; Qingshu Zheng; Zhenxia Chen; Yun Ling*; Yaming ZhouDalton Transactions2019,48(21), 7100-7104 >> Fulltext link

A robust etb-type metal-organic framework showing polarity-exclusive adsorption of acetone over methanol for their azeotropic mixture, Han Hu; Jiaxing Zhu; Feilong Yang; Zhenxia Chen; Mingli Deng; Linhong Weng; Yun Ling*; Yaming ZhouChemical Communications2019,55(46), 6495-6498 >> Fulltext link

   


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